AM251 is a effective CB1 receptor antagonist (IC50/Ki: 8 /7.49 nM) that displays 306-fold selectivity over CB2 receptors, also effective GPR55 agonist (EC50: 39 nM).
Molecular Weight:
555.24
CAS Number:
[183232-66-8]
Formula:
C22H21Cl2IN4O
Target:
Cannabinoid Receptor|||GPR
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