Filgotinib (GLPG0634) is a selective JAK1 inhibitor. The IC50 values against JAK1, JAK2, JAK3, and TYK2 are 10 nM, 28 nM, 810 nM, and 116 nM, respectively.
Molecular Weight:
425.5
CAS Number:
[1206161-97-8]
Formula:
C21H23N5O3S
Target:
JAK|||Tyrosine Kinases
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