AZ31 is an ATM inhibitor with potency, high selectivity, and oral activity.AZ31 inhibits ATM enzymes, intracellular ATM, with IC50 values of <1.2 nM and 46 nM, respectively.AZ31 exhibits excellent ATR selectivity, PIKK family selectivity, and pan-kinase
Molecular Weight:
420.5
CAS Number:
[2088113-98-6]
Formula:
C24H28N4O3
Target:
ATM/ATR
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