Difelikefalin TFA is a kappa-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM
Molecular Weight:
1021.92
CAS Number:
[2742623-88-5]
Formula:
C42H56F9N7O12
Target:
Others
T69530
T69530
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