Difelikefalin HCl is a kappa-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM
Molecular Weight:
789.237
CAS Number:
[2711717-77-8]
Formula:
C36H53N7O6.xHCl
Target:
Others
T69537
T69537
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