Antalarmin is a selective and potent corticotropin-releasing factor receptor 1 (CRHR1) antagonist that crosses the blood-brain barrier and blocks CRF activation and carrageenan-induced subcutaneous inflammation in rats.
Molecular Weight:
378.55
CAS Number:
[157284-96-3]
Formula:
C24H34N4
Target:
CRFR
T70433
T70433
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