Upadacitinib is a potent and selective JAK inhibitor. Upadacitinib is approximately 74 fold selective for Jak1 over Jak2 in cellular assays dependent on specific, relevant cytokines. Upadacitinib demonstrates efficacy in rat arthritis models.
Molecular Weight:
602.521
CAS Number:
[1607431-21-9]
Formula:
C21H33F3N6O11
Target:
ABT-494 , ABT494 , ABT 494
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