BRD4 Inhibitor-28 (Compound 18), an orally active molecule, selectively inhibits the bromodomains of BRD4 (BRD4-BD1 and BRD4-BD2) with IC50 values of 15 and 55 nM, respectively. It also demonstrates inhibition of BRD2-BD1, BRD3-BD1, and BRDT-BD1 with IC5
Molecular Weight:
387.43
CAS Number:
[2468960-80-5]
Formula:
C23H21N3O3
Target:
Epigenetic Reader Domain
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