GSK737 is a dual inhibitor of BRD4 BD1 and BD2, exhibiting pIC50 values of 5.3 and 7.3, respectively. It demonstrates low clearance, along with favorable solubility and permeability in rats [1].
Molecular Weight:
363.41
CAS Number:
[2748687-95-6]
Formula:
C20H21N5O2
Target:
Epigenetic Reader Domain
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