WM-586 is a covalent inhibitor of WDR5 that impedes the WDR5-MYC binding. It selectively reduces the interaction between WDR5 and MYC with an IC50 value of 101 nM, as determined by the HTRF assay [1].
Molecular Weight:
467.47
CAS Number:
[2894832-05-2]
Formula:
C20H20F3N5O3S
Target:
Histone Methyltransferase
* VAT and and shipping costs not included. Errors and price changes excepted