BET-IN-15 (compound 1) is a potent, orally active inhibitor of BET, demonstrating inhibitory IC50 values of 0.64 nM for BRD4-BD1 and 0.25 nM for BRD4-BD2. It exhibits antiproliferative activity [1].
Molecular Weight:
444.45
CAS Number:
[2408994-22-7]
Formula:
C21H18F2N4O3S
Target:
Epigenetic Reader Domain
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