Antitumor agent-101 is a selective, covalent inhibitor targeting lysine methyltransferases G9a/GLP, demonstrating IC50 values of 8.5 nM for G9a and 5.5 nM for GLP. It exhibits antitumor efficacy in the PANC-1 xenograft model [1].
Molecular Weight:
482.62
CAS Number:
[2848632-52-8]
Formula:
C26H38N6O3
Target:
Histone Methyltransferase
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