Selective NaV1.7 channel blocker. Preferentially inhibits neuronal NaV1.7, 1.2 and 1.3 (IC50 values are 26, 150 and 338 nM respectively), compared to muscle subtypes NaV1.4 and 1.5 (IC50 = >10 µM). Inhibits the channel by binding at the neurotoxin recept
Molecular Weight:
4106.79
CAS Number:
[526224-73-7]
Formula:
C174H278N52O51S6
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