Potent and selective µ opioid receptor antagonist (Ki values are 0.96 and >10,000 nM for µ and delta receptors respectively). Causes behavioral effects on central administration in vivo. Also increases K+ currents in rat locus ceruleus neurons in vitro via a
Molecular Weight:
1062.28
CAS Number:
[103429-31-8]
Formula:
C50H67N11O11S2
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