AKAP disruptor. Selectively binds PKA-RI with high affinity (KD values are 6.2 and 12.1 nM for the RIalpha and beta subunits, respectively) and blocks its interaction with AKAP. Inhibits type I PKA-mediated phosphorylation in live cells. Cell permeable.
Molecular Weight:
2401.75
CAS Number:
[TP2129]
Formula:
C109H181N25O35
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